含RGD序列假肽及其模拟物的合成研究概况
STUDY ON THE SYNTHESIS OF RGD-CONTAINING PSEUDOPEPTIDE AND PEPTIDOMIMETICS
作者：杨大成,杨宇,肖晴,钟裕国
Author：
收稿日期： 年卷（期）页码：2001,(06):-440-443
期刊名称：华西药学杂志
Journal Name：WEST CHINA JOURNAL OF PHARMACEUTICAL SCIENCES
关键字：RGD;假肽;肽模拟物;合成;综述
Key words：
基金项目：
中文摘要
通过文献检索 ,综述含RGD序列假肽及肽模拟物的合成研究概况
参考文献
1 PierschbacherMDandRuoslahtiE .Cellattachmentactivityoffibronectincanbeduplicatedbysmallsyntheticfragmentsofthemolecule[J].Na ture,1984,309:30
2 HaymanEG ,PierschbacherMD ,RuolslahtiE .Detachmentofcellsfromculturesubstratebysolublefibronectinpeptide[J].JCellBiol,1985,100(6):1948
3 HynesRO .Afamilyofcellsurfacereceptors[J].Cel1,1987,48:549
4 孙迎庆,郭雁,茹炳根.含RGD的配基与其受体相互作用研究进展[J].生物化学与生物物理进展,1997,24(2):121
5 FujiiH ,NishikawaN ,KomazawaH ,etal.InhibitionoftumorinvasionandmetastasisbypeptidemimeticsofArgGlyAsp(RGD)derivedfromthecellrecognitionsiteoffibronectin[J].OncolRes,1996,8(9):333
6 FujiiH ,NishikawaN ,KomazawaH ,etal.Anewpseudo peptideofArgGlyAsp(RGD)witinhibitoryeffectontumormetastasisandenzy maticdegradationofextracellularmatrix[J].ClinExpMetastasis,1998,16:94
7 LieBL ,IwahoriA ,SampeR ,etal.Synthesisandbiologicalactivityoffourkindsofreversedpeptides[J].BiolPharmBull,1996,19(2):1602
8 MarchandBrynaertJ,DetraitE ,NoisetO ,etal.BiologicalevaluationofRGDpeptidomimetics,designedforthecovalentderivatizationofcellculturesubstrata,aspotentialpromotorsofcellularadhesion[J].Bioma terials,1999,20:1773
9 CarronCP ,MeyerDM ,PeggJA ,etal.Apeptidomimeticantagonistoftheintegrinαvβ3inhibitsLeydigcelltumorgrowthandthedevelopmentof’hypercalcemiaofmalignancy[J].CancerRes,1998,58:1930
10CallahanJ ,BeanJW ,BurgessJL ,etal.DesignandsynthesisofaC7mimeticforthepredictedγ turnconformationfoundinseveralconstrainedRGDantagonists[J].JMedChem,1992,35:3970
11TioengFS ,AdamsSP[P].USPatentApplication,No.4,879,313,Nov7,1989
12AligL ,EdenhoferA ,HadvaryP ,etal.Lowmolecularweight,non peptidefibrinogenreceptorantagonists[J].JMedChem,1992,35,4393
13MarguerieGA ,PlowEF ,EdgingtonTSHumanplateletspossessanin ducibleandsaturablereceptorspecificforfibrinogen[J].JBiolChem,1979,254,5357
14HirschmannR ,NicolaouKC ,PietraicoS ,etal.Nonpeptidalpep tidomimeticswithaβD$Cglucosescaffolding.Apartialsomatostatinag onistbearingaclosestructuralrelationshiptoapotent,selectivesubstancePantagonist[J].JAmChem.Soc,1992,114:9217
15HirschmannR ,SprengelerPA ,KawasakiT ,etal.Theversatilesteroidnucleus:designandsynthesisofapeptidomimeticemployingthisnovelscaffold[J].Tetrahedron,1993,49(17):3665
16HirschmannR ,SprengelerP ,KawasakiT ,etal.Thefirstdesignandsynthesisofasteroidalpeptidomimetic.Thepotentialvalueofpep tidomimeticsinelucidatingthebioactiveconformationofpeptideligands[J].J.Am.Chem.Soc,1992,114:9699
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