吲哚并[3,2-c]喹啉衍生物的微波辅助合成
Microwave irradiation assisted synthesis of indolo [3,2-c] quinoline derivatives
作者:张稳稳;周忠华;曾红;何菱;
Author:
收稿日期: 年卷(期)页码:2008,(03):-263-264
期刊名称:华西药学杂志
Journal Name:WEST CHINA JOURNAL OF PHARMACEUTICAL SCIENCES
关键字:微波辅助合成;Michael加成;Fischer吲哚合成;吲哚并[3,2-c]喹啉;β-苯基萘型化合物
Key words:
基金项目:
中文摘要
目的合成吲哚并[3,2-c]喹啉衍生物并优化其工艺。方法微波辅助Michael加成、环合、Fischer吲哚合成。结果合成了6个吲哚并[3,2-c]喹啉衍生物。结论微波能缩短反应时间,提高Michael加成和Fischer吲哚合成反应的收率。
参考文献
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